商品名:Lipitor, 抑脂妥
Inhibits HMG-CoA reductase, the rate-limiting enzyme in hepatic cholesterol synthesis. Upregulates LDL-receptor activity. Also exerts anti-inflammatory and cardioprotective effects (pleiotropic effects).
Off-label for refractory hyperlipidemia in dogs (dietary management is first-line). Investigational for CHF (anti-inflammatory effects). Also studied for hyperadrenocorticism-associated hyperlipidemia
劑量數字暫停提供:VetPro 的劑量改依 DRUGAPI 藥物資料庫對外的內容,DRUGAPI 目前不提供可直接計算的劑量。下方列出 DRUGAPI 的審查結論與劑量審查引用的來源;計算機可手動輸入劑量換算。
本輪只接受身分、研究族群、標籤與安全界線;所有動物研究數值均留在不可執行證據卡,犬貓計算、處方與自動交互作用維持關閉。
依出現頻率分組;嚴重副作用獨立列出,臨床上需立即辨識。